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Publications:

  1. Jeon, H.; Kim, D.; Lee, J-H.; Song, J.; Lee, W-S.; Kang, D-W.; Kang, S.; Lee, S-B.; Choi, S.; Hong, K-B.; “Hypervalent Iodine-Mediated Alkene Functionalization: Oxazoline and Thiazoline Synthesis via Inter-/Intramolecular Aminohydroxylation and Thioamination”, Advanced Synthesis & Catalysis, (2018), 360, 779

  2. Jang, J.; Kang, D-W.; “Synthesis of Rhamnazin and Ombuin as Methylated Metabolites of Quercetin”, Journal of the Korean Chemical Society, (2018), 62, 19

  3. Ha, H-J.; Kang, D-W.; Kim, H-M.; Kang, J-M.; Ahn, J.; Hyun, H-J.; Lee, J-H.; Kim, S-H.; Kim, H.; Choi, K.; Hong, H-S.; Kim, Y-H.; Jo, D-G.; Lee, J.; Lee, J.; “Discovery of an Orally Bioavailable Benzofuran Analogue That Serves as a β‑Amyloid Aggregation Inhibitor for the Potential Treatment of Alzheimer’s Disease”, Journal of Medicinal Chemistry, (2018), 61, 396

  4. Kang, D-W.; Park, C-S.; “Characterization of Cellulase from Bacillus sp. TH1 Isolated from Environmental Soil”, J. Chitin Chitosan, (2017), 22(3), 156

  5. Lee, E-K.; Park, S-A.; Woo, H.; Park, K. H.; Kang, D-W.; Lim, H.; Kim, Y-T.; “Platinum single atoms dispersed on carbon nanotubes as reusable catalyst for Suzuki coupling reaction”, Journal of Catalysis, (2017), 352, 388   발행년월일 2017-

  6. Lee, S.; Kang, D-W.; Ryu, H.; Kim, C.; Ahn, J.; Lee, H.; Kim, E.; Hong, S.; Choi, S; Blumberg, P. M.; Frank-Foltyn, R.; Bahrenberg, G.; Stockhausen, H.; Christoph, T.; Lee, J.; “t-Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists”, Bioorganic & Medicinal Chemistry, (2017), 25, 2451    발행년월일 2017-03-06      ISSN 0968-0896

  7. Ahn, J.; Jung, A.; Kim, M-Y.; Kim, H-M.; Ryu, H.; Kim, S.; Kang, D-W.; Hong, S.; Cui, M.; Choi, S.; Blumberg, P. M.; Frank-Foltyn, R.; Bahrenberg, G.; Stockhausen, H.; Christoph, T.; Lee, J.; “Structure activity relationships of benzyl C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists”, Bioorganic & Medicinal Chemistry, (2015), 23, 6844  발행년월일 2015-10-09      ISSN 0968-0896

  8. Ryu, H.; Seo, S.; Cho, S-H.; Kim H. S.; Jung, A.; Kang, D-W.; Son, K.; Cui, M.; Hong, S-H.; Sharma, P. K.; Choi, S.; Blumberg, P. M.; Frank-Foltyn, R.; Bahrenberg, G.; Stockhausen, H.; Schiene, K.; Christoph, T.; Frormann, S.; Lee, J.; “2-Alkyl/alkenyl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists” Bioorganic & Medicinal Chemistry Letters, (2014), 24, 4039   발행년월일 2014-06-02      ISSN 0960-894X

  9. Kim, E. J.; Abramowitz, L. K.; Bond, M. R.; Love, D. C.; Kang, D-W.; Luecke, H. F.; Kang, D. W.; Ahn, J-S.; Hanover, J. A.;  “Versatile O-GlcNAc Transferase Assay for High-Throughput Identification of Enzyme Variants, Substrates, and Inhibitors” Bioconjugate Chemistry, (2014), 25, 1025 발행년월 2014-05-27         ISSN 1043-1802

  10. Kang, D-W.; Kim, E. J.; “Design, Synthesis and Preliminary Biological Evaluation of a Biotin-S-S-Phosphine Reagent” Bull. Korean Chem. Soc., (2014), 35(2), 383     발행년월 2014-02             ISSN 0253-2964

  11. Kang, D-W.; “Synthesis of Glucuronic Acid Conjugates of Linoleic Acid Metabolites” Journal of the Korean Chemical Society, (2013), 57(6), 738         발행년월 2013-12             ISSN 1017-2548

  12. Sakakibara, N.; Chen, D.; Jang, M. K.; Kang, D-W.; Luecke, H. F.; Wu, S. Y.; Chiang, C.-M.; McBride, A. A; “Brd4 Is Displaced from HPV Replication Factories as They Expand and Amplify Viral DNA” PLOS Pathogens, (2013), 9(11), e1003777      발행년월 2013-11             ISSN 1553-7366

  13. Johnson, C. H.; Bonzo, J. A.; Cheng, J.; Krausz, K. W.; Kang, D-W.; Luecke, H.; Idle, J. R.; Gonzalez, F. J.; “Cytochrome P450 Regulation by alpha-Tocopherol in Pxr-Null and PXR-Humanized Mice” Drug Metabolism and Disposition, (2013), 41, 406       발행년월 2013-11             ISSN 1521-009X

  14. Kang, D-W.; Hans F. Luecke; “Facile Synthetic Routes to Prepare alpha-Muricholic Acid, Hyocholic Acid, and Their Taurine Conjugates” Bull. Korean Chem. Soc., (2013), 34(8), 2436           발행년월 2013-08          ISSN 0253-2964

  15. Kim, E. J.; Kang, D-W.; Luecke, H. F.; Bond, M. R.; Ghosh, S.; Love, D. C.; Ahn, J-S.; Kang, D-O; Hanover, J. A.; “Optimizing the selectivity of DIFO-based reagents for intracellular bioorthogonal applications” Carbohydrate Research, (2013), 377, 18           발행년월 2013-08             ISSN 0008-6215

  16. Thorat, S. A.; Kang, D-W.; Ryu, H.; Kim, M-S.; Kim, H-S.; Ann, J.; Ha, T.; Kim, S-E.; Son, K.; Choi, Sun; Blumberg, P. M.; Frank, R.; Bahrenberg, G.; Schiene, K.; Christoph, T.; Lee, J.; “2-(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists: Structure activity relationship of the 2-oxy pyridine C-region” European Journal of Medicinal Chemistry, (2013), 64, 589           발행년월 2013-06 ISSN 0223-5234

  17. Matsubara, T.; Tanaka, N.; Krausz, K. W.; Manna, S. K.; Kang, D-W.; Anderson, E. R.; Luecke, H.; Patterson, A. D.; Shah, Y. M.; Gonzalez, F. J.; “Metabolomics identifies an inflammatory cascade involved in dioxin- and diet-induced steatohepatitis” Cell Metabolism, (2012), 16(5), 634      발행년월 2012-11-07  ISSN 1550-4131

  18. Matsubara, T.; Tanaka, N.; Sato, M.; Kang, D-W.; Krausz, K. W.; Flanders, K. C.; Ikeda, K.; Luecke, H.; Wakefield, L. M.; Gonzalez, F. J.; “TGF-b-SMAD3 signaling mediates hepatic bile acid and phospholipid metabolism following lithocholic acid-induced liver injury” J. Lipid Research, (2012), 53(12), 2698     발행년월일 2012-10-03         ISSN 0022-2275

  19. Johnson, C. H.; Patterson, A. D.; Krausz, K. W.; Kalinich, J. F.; Tyburski, J. B.; Kang, D-W.; Luecke, H.; Gonzalez, F. J.; Blakely, W. F.; Idle, J. R.; “Radiation Metabolomics. 5. Identification of urinary biomarkers of ionizing radiation exposure in nonhuman primates by mass spectrometry-based metabolomics” Radiation Research, (2012), 178, 328           발행년월 2012-10 ISSN 0033-7587

  20. Johnson, C. H.; Slanar, O.; Krausz, K. W.; Kang, D-W.; Patterson, A. D.; Kim, J-H.; Luecke, H.; Gonzalez, F. J.; Idle, J. R.; “Novel metabolites and roles for a-tocopherol in humans and mice discovered by mass spectrometry-based metabolomics” Am. J. Clin. Nutr., (2012), 96, 818      발행년월 2012-10-01         ISSN 0002-9165

  21. Kim, M-S.; Ryu, H.; Kang, D-W.; Kim, H-S.; Cho, S-H.; Seo, S.; Park, Y-S.; Kim, M-Y.; Kwak, E-J.; Kim, Y-S.; Bhondwe, R. S.; Kim, H-S.; Park, S-G.; Son, K.; Choi, S.; DeAndrea-Lazarus, I. A.; Pearce, L. V.; Blumberg, P. M.; Frank, R.; Bahrenberg, G.; Stockhausen, H.; Kogel, B. Y.; Schiene, K.; Christoph, T.; Lee, J.; “2-(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as potent transient receptor potential vanilloid 1 (TRPV1) antagonists: structure-activity relationships of 2-amino derivatives in the N-(6-trifluoromethylpyridin-3-ylmethyl) C-region” Journal of Medicinal Chemistry, (2012), 55, 8392     발행년월일 2012-10-11       ISSN 0022-2623

  22. Bhondwe, R. S.; Kang, D-W.; Kim, M-S.; Kim, H-S.; Park, S-G.; Son, K.; Choi, S.; Kuhs, K. A. L.; Pavlyukovets, V. A.; Pearce, L. V.; Blumberg, P. M.; Lee, J.; “Structure-activity relationships and molecular modeling of the N-(3-pivaloyloxy-2-benzylpropyl)-N’-[4-(methylsulfonylamino)benzyl]thiourea template for TRPV1 antagonism” Bioorganic & Medicinal Chemistry Letters, (2012), 22, 3656   발행년월일 2012-06-01      ISSN 0960-894X

  23. Sun, W.; Liu, K.; Ryu, H.; Kang, D-W.; Kim, Y-S.; Kim, M-S.; Cho, Y.; Bhondwe, R. S.; Thorat, S. A.; Kim H-S.; Pearce, L. V.; Pavlyukovets, V. A.; Tran, R.; Morgan, M. A.; Lazar, J.; Ryder, C. B.; Toth, A.; Blumberg, P. M.; Lee, J.; “2-(4-Methylsulfonylaminophenyl)propanamide TRPV1 antagonists: Structure-activity relationships in the B and C-regions” Bioorganic & Medicinal Chemistry, (2012), 20, 1310 발행년월일 2013-01-01      ISSN 0968-0896

  24. Lee, J-H.; Lee, Y.; Ryu, H.; Kang, D-W.; Lee, J.; Lazar, J.; Pearce, L. V.; Pavlyukovets, V. A.; Blumberg, P. M.; Choi, S.; “Structural insights into transient receptor potential vanilloid type 1 (TRPV1) from homology modeling, flexible docking, and mutational studies” J. Computer-Aided Molecular Design, (2011), 25(4), 317       발행년월 2011-04          ISSN 0920-654X

  25. Johnson, C. H.; Patterson, A. D.; Krausz, K. W.; Lanz, C.; Kang, D-W.; Luecke, H.; Gonzalez, F. J.; Idle, J. R.; “Radiation Metabolomics. 4. UPLC-ESI-QTOFMS-Based metabolomics for urinary biomarker discovery in gamma-irradiated rats” Radiation Research, (2011), 175, 473     발행년월 2011-04   ISSN 0033-7587

  26. Lim, K-S.; Kang, D-W.; Kim, Y-S.; Kim, M-S.; Park, S-G.; Choi, S.; Pearce, L. V.; Blumberg, P. M.; Lee, J.; “Receptor activity and conformational analysis of 5’-halogenated resiniferatoxin analogues as TRPV1 ligands” Bioorganic & Medicinal Chemistry Letters, (2011), 21(1), 299 발행년월일 2011-01-01      ISSN 0960-894X

  27. Kang, D-W.; Kim, Y-S.; Lim, K-S.; Kim, M-S.; Pearch, L. V.; Pavlyukovets, V. A.; Tao, A. K.; Lang-Kuhs, K. A.; Blumberg, P. M.; Lee, J.; “Halogenation of 4-hydroxy/amino-3-methoxyphenyl acetamide TRPV1 agonists showed enhanced antagonism to capsaicin” Bioorganic & Medicinal Chemistry, (2010), 18(22), 8092         발행년월일 2010-11-15          ISSN 0968-0896

  28. Cho, J-Y.; Matsubara, T.; Kang, D-W.; Ahn, S-H.; Krausz, K. W.; Idle, J. R.; Luecke, H.; Gonzalez, F. J.; “Urinary metabolomics in Fxr-null mice reveals activated adaptive metabolic pathways upon bile acid challenge.” J. Lipid Research, (2010), 51(5), 1063     발행년월일 2010-11-09            ISSN 0022-2275

  29. Tosh, D. K.; Chinn, M.; Yoo, L. S.; Kang, D-W.; Luecke, H.; Gao, Z-G.; Jacobson, K. A.; “2-Dialkynyl derivatives of (N)-methanocarba nucleosides: ‘Clickable’ A3 adenosine receptor-selective agonists” Bioorganic & Medicinal Chemistry, (2010), 18(2), 508      발행년월일 2010-01-15      ISSN 0968-0896

  30. Cho, J-Y.; Kang, D-W.; Ma, X.; Ahn, S-H.; Krausz, K. W.; Luecke, H.; Idle, J. R.; Gonzalez, F. J.; “Metabolomics reveals a novel vitamin E metabolite and attenuated vitamin E metabolism upon PXR activation” J. Lipid Research, (2009), 50(5), 924       발행년월일 2009-01-13           ISSN 0022-2275

  31. Choi, H-K.; Choi, S.; Lee, Y.; Kang, D-W.; Ryu, H.; Maeng, H-J.; Chung, S-J.; Pavlyukovets, V. A.; Pearce, L. V.; Toth, A.; Tran, R.; Wang, Y.; Morgan, M. A.; Blumberg, P. M.; Lee, J.; “Non-vanillyl resiniferatoxin analogues as potent and metabolically stable transient receoptor potential vanilloid 1 agonists” Bioorganic & Medicinal Chemistry, (2009), 17(2), 690      발행년월일 2009-01-15      ISSN 0968-0896

  32. Lim, J-O.; Jin, M-K.; Ryu, H.; Kang, D-W.; Lee, J.; Pearce, L. V.; Tran, R.; Toth, A.; Blumberg, P. M.; “Conformationally constrained analogues of N’-(4-tert-butylbenzyl)-N-(4-methylsulfonylamonobenzyl)thiourea as TRPV1 antagonists” European J. Medicinal Chemistry, (2009), 44(1), 322       발행년월 2009-01 ISSN 0223-5234

  33. Pearce, L. V.; Toth, A.; Ryu, H.; Kang, D-W.; Choi, H-K.; Jin, M-K.; Lee, J.; Blumberg, P. M.; “Differential modulation of agonist and antagonist structure activity relations for rat TRPV1 by cyclosporine A and other protein phosphatase inhibitors” Naunyn-Schmiedeberg’s Archives of Pharmacology, (2008), 377(2), 149    발행년월 2008-04          ISSN 0028-1298

  34. Ryu, H.; Jin, M-K.; Kim, S-Y.; Choi, H-K.; Kang, S-U.; Kang, D-W.; Lee, J.; Pearce, L. V.; Pavlyukovets, V. A.; Morgan, M. A.; Tran, R.; Toth, A.; Lundberg, D. J.; Blumberg, P. M.; “Stereospecific high-affinity TRPV1 antagonists: Chiral N-(2-Benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide analogues” J. Medicinal Chemistry, (2008), 51(1), 57  발행년월일 2007-12-12      ISSN 0022-2623

  35. Buckheit, R. W. Jr.; Hartman, T. L.; Watson, K. M.; Kwon, H-S.; Lee, S-H.; Lee, J-W.; Kang, D-W.; Chung, S-G.; Cho, E-W.; “The structure-activity relationships of 2,4-(1H,3H)-pyrimidinedione derivatives as potent HIV type 1 and type 2 inhibitors” Antiviral Chemistry & Chemotherapy, (2007), 18(5), 259  발행년월 2017-05 ISSN 0956-3202

  36. Chung, J-U.; Kim, S-Y.; Lim, J-O.; Choi, H-K.; Kang, S-U.; Yoon, H-S.; Ryu, H.; Kang, D-W.; Lee, J.; Kang, B.; Choi, S.; Toth, A.; Pearce, L. V.; Pavlyukovets, V. A.; Lundberg, D. J.; Blumberg, P. M.; “a-Substituted N-(4-tert-butylbenzyl)-N’-[4-methylsulfonylamino]benzyl]thiourea analogues as petent and stereospecific TRPV1 antagonists” Bioorganic & Medicinal Chemistry, (2007), 15(18), 6043         발행년월일 2007-09-15      ISSN 0968-0896

  37. Kang, D-W.; Ryu, H.; Lee, J.; Lang, K. A.; Pavlyukovets, V. A.; Pearce, L. V.; Ikeda, T.; Lazar J.; Blumberg, P. M.; “Halogenation of 4-hydroxy-3-methoxybenzyl thiourea TRPV1 agonists showed enchanced antagonism to capsaicin” Bioorganic & Medicinal Chemistry Letters, (2007), 17(1), 214           발행년월일 2007-01-01         ISSN 0960-894X

  38. Yi, E-Y.; Jeong, E-J.; Kang, D-W.; Joo, J-H.; Kwon, H-S.; Lee, S-H.; Park, S-K.; Chung, S-G.; Cho, E-H.; Kim, Y-J.; “Anti-angiogenic and anti-tumor apoptotic activities of a topoisomerase II inhibiting agent SJ-8026” International J. Oncology, (2005), 26(6), 1613     발행년월 2005-06       ISSN 1019-6439

  39. Yi, E-Y.; Jeong, E-J.; Song, H-S.; Lee, M-S.; Kang, D-W.; Joo, J-H.; Kwon, H-S.; Lee, S-H.; Park, S-K.; Chung, S-G.; Cho, E-H.; Kim, Y-J.; “Anti-angiogenic and anti-tumor apoptotic activities of SJ-8002, a new piperazine derivative” International J. Oncology, (2004), 25(2), 365          발행년월 2004-08   ISSN 1019-6439

  40. Lee, J-H.; Kang, D-W.; Kwon, H-S.; Lee, S-H.; Park, S-K.; Chung, S-G.; Cho, E-H.; Paik, S-Y.; Lee, J-H.; “Microtube inhibitory effects of various SJ compounds on tissue culture cells” Archives of Pharmacal Research, (2004), 27(4), 436      발행년월 2004-04         ISSN 0253-6269

  41. Lee, Y-S.; Kang, D-W.; Lee, S-J.; Park, H.; “Asymmetric synthesis of both enantiomers of pyrrolidinoisoquinoline derivatives from L-malic acid and L-tartaric acid” J. Organic Chemistry, (1995), 60(22), 7149  발행년월 1995-11        ISSN 0022-3263

  42. Lee, Y-S.; Kang, D-W.; Lee, S-J.; Park, H.; “Stereoselective synthesis of an isoquinolidinone by acyliminium ion cyclization of chiral hydroxylactams” Synthetic Communications, (1995), 25(13), 1947   발행년월 1995-07     ISSN 0039-7911

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